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1

Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine

Piekielna, Justyna, Gentilucci, Luca, De Marco, Rossella, Perlikowska, Renata, Adamska, Anna, Olczak, Jacek, Mazur, Marzena, Artali, Roberto, Modranka, Jakub, Janecki, Tomasz, Tömböly, Csaba, Janecka,

Journal:

Bioorganic & Medicinal Chemistry

Year:

2014

Language:

english

File:

PDF, 970 KB

english, 2014

2

Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration

Perlikowska, Renata, Piekielna, Justyna, Gentilucci, Luca, De Marco, Rossella, Cerlesi, Maria Camilla, Calo, Girolamo, Artali, Roberto, Tömböly, Csaba, Kluczyk, Alicja, Janecka, Anna

Journal:

European Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 849 KB

english, 2015

3

Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic

Piekielna, Justyna, De Marco, Rossella, Gentilucci, Luca, Cerlesi, Maria Camilla, Calo', Girolamo, Tömböly, Csaba, Artali, Roberto, Janecka, Anna

Journal:

Year:

2016

Language:

english

File:

PDF, 345 KB

english, 2016

4

Synthesis and Evaluation of the β-Turn Properties of 4-Amino-1,2,4,5-tetrahydro-2-benzazepin-3-ones and of Their Spirocyclic Derivative

Karolien Van Rompaey, Steven Ballet, Csaba Tömböly, Rien De Wachter, Kenno Vanommeslaeghe, Monique Biesemans, Rudolph Willem, Dirk Tourwé

Journal:

European Journal of Organic Chemistry

Year:

2006

Language:

english

File:

PDF, 246 KB

english, 2006

5

Preparation of specifically tritiated endomorphins

Csaba Tömböly, Rajiv Dixit, Imre Lengyel, Anna Borsodi, Géza Tóth

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2001

File:

PDF, 1.52 MB

2001

6

Liquid chromatographic study of the enzymatic degradation of endomorphins, with identification by electrospray ionization mass spectrometry

Antal Péter, Géza Tóth, Csaba Tömböly, Georges Laus, Dirk Tourwè

Journal:

Journal of Chromatography A

Year:

1999

Language:

english

File:

PDF, 191 KB

english, 1999

7

Effects of endomorphin-1 on open-field behavior and on the hypothalamic-pituitary-adrenal system

Erika Bujdosó, Miklós Jászberényi, Csaba Tömböly, Géza Tóth, Gyula Telegdy

Journal:

Endocrine (Springer)

Year:

2001

Language:

english

File:

PDF, 77 KB

english, 2001

8

Specific activation of the μ opioid receptor (MOR) by endomorphin 1 and endomorphin 2

Krisztina Monory, Marie-Claude Bourin, Mariana Spetea, Csaba Tömböly, Géza Tóth, Hans W. Matthes, Brigitte L. Kieffer, Jacques Hanoune, Anna Borsodi

Journal:

European Journal of Neuroscience

Year:

2000

Language:

english

File:

PDF, 269 KB

english, 2000

9

In VitroBinding and Signaling Profile of the Novel μ Opioid Receptor Agonist Endomorphin 2 in Rat Brain Membranes

Mariana Spetea, Krisztina Monory, Csaba Tömböly, Géza Tóth, Eleni Tzavara, Sándor Benyhe, Jacques Hanoune, Anna Borsodi

Journal:

Biochemical and Biophysical Research Communications

Year:

1998

Language:

english

File:

PDF, 120 KB

english, 1998

10

Influence of Degradation on Binding Properties and Biological Activity of Endomorphin 1

Ildikó Szatmári, Dauren Biyashev, Csaba Tömböly, Géza Tóth, Mónika Mácsai, Gyula Szabó, Anna Borsodi, Imre Lengyel

Journal:

Biochemical and Biophysical Research Communications

Year:

2001

Language:

english

File:

PDF, 74 KB

english, 2001

11

Selective and high affinity labeling of neuronal and recombinant nociceptin receptors with the hexapeptide radioprobe [3H]Ac-RYYRIK-ol

Engin Bojnik, Judit Farkas, Anna Magyar, Csaba Tömböly, Ümit Güçlü, Özge Gündüz, Anna Borsodi, Maïthe Corbani, Sándor Benyhe

Journal:

Neurochemistry International

Year:

2009

Language:

english

File:

PDF, 711 KB

english, 2009

12

Autoradiography in opioid triple knockout mice reveals opioid and opioid receptor like binding of naloxone benzoylhydrazone

Veronica Cox, Siân Clarke, Tracy Czyzyk, Micheal Ansonoff, Joshua Nitsche, Ming-Sing Hsu, Anna Borsodi, Csaba Tömböly, Géza Tóth, Ray Hill, John Pintar, Ian Kitchen

Journal:

Neuropharmacology

Year:

2005

Language:

english

File:

PDF, 1.41 MB

english, 2005

13

Endomorphin-1 and endomorphin-2 differentially interact with specific binding sites for substance P (SP) aminoterminal SP1–7 in the rat spinal cord

Milad Botros, Mathias Hallberg, Tobias Johansson, Qin Zhou, Gunnar Lindeberg, Per-Anders Frändberg, Csaba Tömböly, Géza Tóth, Pierre Le Grevès, Fred Nyberg

Journal:

Year:

2006

Language:

english

File:

PDF, 156 KB

english, 2006

14

Endomorphins interact with the substance P (SP) aminoterminal SP1–7 binding in the ventral tegmental area of the rat brain

Milad Botros, Tobias Johansson, Qin Zhou, Gunnar Lindeberg, Csaba Tömböly, Géza Tóth, Pierre Le Grevès, Fred Nyberg, Mathias Hallberg

Journal:

Year:

2008

Language:

english

File:

PDF, 185 KB

english, 2008

15

Antinociceptive effects of intrathecal endomorphin-1 and -2 in rats

Gyöngyi Horvath, Margit Szikszay, Csaba Tömböly, György Benedek

Journal:

Year:

1999

Language:

english

File:

PDF, 538 KB

english, 1999

16

In vitro quantitative study of the degradation of endomorphins

Csaba Tömböly, Antal Péter, Géza Tóth

Journal:

Year:

2002

Language:

english

File:

PDF, 202 KB

english, 2002

17

β-Methyl Substitution of Cyclohexylalanine in Dmt-Tic-Cha-Phe Peptides Results in Highly Potent δ Opioid Antagonists

Tóth, Géza, Ioja, Enikő, Tömböly, Csaba, Ballet, Steven, Tourwé, Dirk, Péter, Antal, Martinek, Tamás, Chung, Nga N., Schiller, Peter W., Benyhe, Sándor, Borsodi, Anna

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 66 KB

english, 2007

18

Preparation of Semisynthetic Lipoproteins with Fluorescent Cholesterol Anchor and Their Introduction to the Cell Membrane with Minimal Disruption of the Membrane

Schäfer, Balázs, Orbán, Erika, Borics, Attila, Huszár, Krisztina, Nyeste, Antal, Welker, Ervin, Tömböly, Csaba

Journal:

Bioconjugate Chemistry

Year:

2013

Language:

english

File:

PDF, 3.68 MB

english, 2013

19

In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt 1 -DALDA Analogues

Ballet, Steven, Betti, Cecilia, Novoa, Alexandre, Tömböly, Csaba, Uhd Nielsen, Carsten, Helms, Hans Christian, Lesniak, Anna, Kleczkowska, Patrycja, Chung, Nga N., Lipkowski, Andrzej W., Brodin, Birge

Journal:

ACS Medicinal Chemistry Letters

Year:

2014

Language:

english

File:

PDF, 675 KB

english, 2014

20

Pharmacological characterization of endomorphin-2-based cyclic pentapeptides with methylated phenylalanine residues

Perlikowska, Renata, Malfacini, Davide, Cerlesi, Maria Camilla, Calo’, Girolamo, Piekielna, Justyna, Floriot, Léonore, Henry, Tiphaine, do-Rego, Jean Claude, Tömböly, Csaba, Kluczyk, Alicja, Janecka,

Journal:

Year:

2014

Language:

english

File:

PDF, 534 KB

english, 2014

21

Unprecedented Sigmatropic Rearrangements Leading to 2,3-Dihydro-1 H -2-benzazepine-3-carboxylic Acid

Martins, José C., Van Rompaey, Karolien, Wittmann, Guyla, Tömböly, Csaba, Tóth, Géza, De Kimpe, Norbert, Tourwé, Dirk

Journal:

Journal of Organic Chemistry

Year:

2001

Language:

english

File:

PDF, 45 KB

english, 2001

22

Endomorphin-2 with a β-Turn Backbone Constraint Retains the Potent μ-Opioid Receptor Agonist Properties

Tömböly, Csaba, Ballet, Steven, Feytens, Debby, Kövér, Katalin E., Borics, Attila, Lovas, Sándor, Al-Khrasani, Mahmoud, Fürst, Zsuzsanna, Tóth, Géza, Benyhe, Sándor, Tourwé, Dirk

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 287 KB

english, 2008

23

Structure−Activity Study on the Phe Side Chain Arrangement of Endomorphins Using Conformationally Constrained Analogues

Tömböly, Csaba, Kövér, Katalin E., Péter, Antal, Tourwé, Dirk, Biyashev, Dauren, Benyhe, Sándor, Borsodi, Anna, Al-Khrasani, Mahmoud, Rónai, András Z., Tóth, Géza

Journal:

Journal of Medicinal Chemistry

Year:

2004

Language:

english

File:

PDF, 90 KB

english, 2004

24

Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines

Piekielna, Justyna, Perlikowska, Renata, do-Rego, Jean Claude, do-Rego, Jean-Luc, Cerlesi, Maria Camilla, Calo, Girolamo, Kluczyk, Alicja, Łapiński, Krzysztof, Tömböly, Csaba, Janecka, Anna

Journal:

ACS Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 470 KB

english, 2015

25

Ring size in cyclic endomorphin-2 analogs modulates receptor binding affinity and selectivity

Piekielna, Justyna, Kluczyk, Alicja, Gentilucci, Luca, Cerlesi, Maria Camilla, Calo’, Girolamo, Tomböly, Csaba, Łapiński, Krzysztof, Janecki, Tomasz, Janecka, Anna

Journal:

Organic & Biomolecular Chemistry

Year:

2015

Language:

english

File:

PDF, 591 KB

english, 2015

26

Semisynthesis of membrane-anchored cholesteryl lipoproteins on live cell surface by azide–alkyne click reaction

Schäfer, Balázs, Orbán, Erika, Fiser, Gabriella, Marton, Annamária, Vizler, Csaba, Tömböly, Csaba

Journal:

Tetrahedron Letters

Year:

2016

Language:

english

File:

PDF, 1.20 MB

english, 2016

27

Investigation of receptor binding and functional characteristics of hemopressin(1–7)

Dvorácskó, Szabolcs, Tömböly, Csaba, Berkecz, Róbert, Keresztes, Attila

Journal:

Year:

2016

Language:

english

File:

PDF, 621 KB

english, 2016

28

Correction for “Synthesis of Mixed Opioid Affinity Cyclic Endomorphin-2 Analogues with Fluorinated Phenylalanines”

Piekielna, Justyna, Perlikowska, Renata, do-Rego, Jean-Claude, do-Rego, Jean-Luc, Cerlesi, Maria Camilla, Calo, Girolamo, Kluczyk, Alicja, Łapiński, Krzysztof, Tömböly, Csaba, Janecka, Anna

Journal:

ACS Medicinal Chemistry Letters

Year:

2016

Language:

english

File:

PDF, 125 KB

english, 2016

29

The Effects of Peptide and Lipid Endocannabinoids on Arthritic Pain at the Spinal Level

Petrovszki, Zita, Kovacs, Gyula, Tömböly, Csaba, Benedek, György, Horvath, Gyongyi

Journal:

Anesthesia & Analgesia

Year:

2012

Language:

english

File:

PDF, 1.90 MB

english, 2012

30

Tritium labelling of a cholesterol amphiphile designed for cell membrane anchoring of proteins

Schäfer, Balázs, Orbán, Erika, Kele, Zoltán, Tömböly, Csaba

Journal:

Journal of Labelled Compounds and Radiopharmaceuticals

Year:

2015

Language:

english

File:

PDF, 512 KB

english, 2015

31

Further Characterization of Hemopressin Peptide Fragments in the Opioid and Cannabinoid Systems

Szlavicz, Eszter, Perera, Pannilage Shiromi, Tomboly, Csaba, Helyes, Zsuzsanna, Zador, Ferenc, Benyhe, Sandor, Borsodi, Anna, Bojnik, Engin

Journal:

Anesthesia & Analgesia

Year:

2015

Language:

english

File:

PDF, 963 KB

english, 2015

32

Decreased CB receptor binding and cannabinoid signaling in three brain regions of a rat model of schizophrenia

Szűcs, Edina, Dvorácskó, Szabolcs, Tömböly, Csaba, Büki, Alexandra, Kékesi, Gabriella, Horváth, Gyöngyi, Benyhe, Sándor

Journal:

Neuroscience Letters

Year:

2016

Language:

english

File:

PDF, 694 KB

english, 2016

33

Cyclic mu-opioid receptor ligands containing multiple N -methylated amino acid residues

Adamska-Bartłomiejczyk, Anna, Janecka, Anna, Szabó, Márton Richárd, Cerlesi, Maria Camilla, Calo, Girolamo, Kluczyk, Alicja, Tömböly, Csaba, Borics, Attila

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2017

Language:

english

File:

PDF, 961 KB

english, 2017

34

Emotional disorders induced by Hemopressin and RVD-hemopressin(α) administration in rats

Leone, Sheila, Recinella, Lucia, Chiavaroli, Annalisa, Martinotti, Sara, Ferrante, Claudio, Mollica, Adriano, Macedonio, Giorgia, Stefanucci, Azzurra, Dvorácskó, Szabolcs, Tömböly, Csaba, De Petrocell

Journal:

Pharmacological Reports

Year:

2017

Language:

english

File:

PDF, 453 KB

english, 2017

35

Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis -4-amino-L-proline residues

Adamska-Bartłomiejczyk, Anna, Borics, Attila, Tömböly, Csaba, Dvorácskó, Szabolcs, Lisowski, Marek, Kluczyk, Alicja, Wołczański, Grzegorz, Piekielna-Ciesielska, Justyna, Janecka, Anna

Journal:

Journal of Peptide Science

Year:

2017

Language:

english

File:

PDF, 365 KB

english, 2017

36

Neuroanatomical distribution and function of the vasopressin V 1B receptor in the rat brain deciphered using specific fluorescent ligands

Corbani, Maithé, Marir, Rafik, Trueba, Miguel, Chafai, Magda, Vincent, Anne, Borie, Amélie M., Desarménien, Michel G., Ueta, Yoichi, Tomboly, Csaba, Olma, Aleksandra, Manning, Maurice, Guillon, Gilles

Journal:

General and Comparative Endocrinology

Year:

2017

Language:

english

File:

PDF, 7.14 MB

english, 2017

37

Development of potent and proteolytically stable human neuromedin U receptor agonists

De Prins, An, Martin, Charlotte, Van Wanseele, Yannick, Skov, Louise Julie, Tömböly, Csaba, Tourwé, Dirk, Caveliers, Vicky, Van Eeckhaut, Ann, Holst, Birgitte, Rosenkilde, Mette Marie, Smolders, Ilse,

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 2.37 MB

english, 2017

38

Effects of central RVD-hemopressin(α) administration on anxiety, feeding behavior and hypothalamic neuromodulators in the rat

Recinella, Lucia, Chiavaroli, Annalisa, Ferrante, Claudio, Mollica, Adriano, Macedonio, Giorgia, Stefanucci, Azzurra, Dimmito, Marilisa Pia, Dvorácskó, Szabolcs, Tömböly, Csaba, Brunetti, Luigi, Orlan

Journal:

Pharmacological Reports

Year:

2018

Language:

english

File:

PDF, 531 KB

english, 2018

39

Synthesis and in vitro evaluation of stabilized and selective Neuromedin U-1 receptor agonists

De Prins, An, Martin, Charlotte, Van Wanseele, Yannick, Tomboly, Csaba, Tourwé, Dirk, Caveliers, Vicky, Holst, Birgitte, Van Eeckhaut, Ann, Rosenkilde, Mette Marie, Smolders, Ilse, Ballet, Steven

Journal:

ACS Medicinal Chemistry Letters

Year:

2018

Language:

english

File:

PDF, 462 KB

english, 2018

40

Interactions between the Kynurenine and the Endocannabinoid System with Special Emphasis on Migraine

Nagy-Grócz, Gábor, Zádor, Ferenc, Dvorácskó, Szabolcs, Bohár, Zsuzsanna, Benyhe, Sándor, Tömböly, Csaba, Párdutz, Árpád, Vécsei, László

Journal:

International Journal of Molecular Sciences

Year:

2017

Language:

english

File:

PDF, 1.17 MB

english, 2017

41

Novel Fubinaca/Rimonabant hybrids as endocannabinoid system modulators

Stefanucci, Azzurra, Macedonio, Giorgia, Dvorácskó, Szabolcs, Tömböly, Csaba, Mollica, Adriano

Journal:

Year:

2018

Language:

english

File:

PDF, 1.73 MB

english, 2018

42

Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13 β - and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis

Bacsa, Ildikó, Herman, Bianka Edina, Jójárt, Rebeka, Herman, Kevin Stefán, Wölfling, János, Schneider, Gyula, Varga, Mónika, Tömböly, Csaba, Rižner, Tea Lanišnik, Szécsi, Mihály, Mernyák, Erzsébet

Journal:

Journal of Enzyme Inhibition and Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 3.44 MB

english, 2018

43

Effects of RVD-hemopressin (α) on feeding and body weight after standard or cafeteria diet in rats

Leone, Sheila, Ferrante, Claudio, Recinella, Lucia, Chiavaroli, Annalisa, Mollica, Adriano, Tömböly, Csaba, Stefanucci, Azzurra, Dimmito, Marilisa Pia, Dvorácskó, Szabolcs, Verratti, Vittore, De Petro

Journal:

Year:

2018

Language:

english

File:

PDF, 674 KB

english, 2018